Cyclazocine

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Cyclazocine
Systematic (IUPAC) name
?
Identifiers
CAS number	?
ATC code	?
PubChem	19143
Chemical data
Formula	C18H25NO
Mol. mass	271.397 g/mol
Pharmacokinetic data
Bioavailability	?
Metabolism	?
Half life	?
Excretion	?
Therapeutic considerations
Pregnancy cat.	?
Legal status
Routes	?

Cyclazocine is a mixed opiate agonist-antagonist related to dezocine, pentazocine and phenazocine. This family of opioid drugs is called the benzomorphans or benzazocines.

[edit] Use

Research into the use of cyclazocine for the treatment of Bipolar patients with depression was undertaken by Fink and colleagues (1970). It showed that 8 out of 10 patients experienced moderate improvement.

Research during the 1960s and 1970s into the possible use of cyclazocine for management of pain, and later for assisting treatment of narcotic addiction was severely hampered by the drug's psychotomimetic, dysphoric, and hallucinatory effects.

[edit] Dosage

Dosages of 1-3mg were administered in the tests

[edit] See also

• Ketazocine

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